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德拉沙星中间体

名称

CAS#

结构式

ethyl 3-(3-chloro-2,4,5-trifluorophenyl)-3-oxopropanoate

101987-86-4

 

2,3,5,6-tetrafluoropyridine

2875-18-5

 

3,5-difluoropyridine-2,6-diamine

247069-27-8

 

3-Hydroxyazetidine hydrochloride

18621-18-6

 

ethyl 1-(6-amino-3,5-difluoropyridin-2-yl)-8-chloro-6-fluoro-7-(3-hydroxyazetidin-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylate

1620905-72-7

 

ethyl 1-(6-amino-3,5-difluoropyridin-2-yl)-8-chloro-6,7-difluoro-4-oxo-1,4-dihydroquinoline-3-carboxylate

189279-51-4

 

ethyl 1-(6-amino-3,5-difluoropyridin-2-yl)-6-fluoro-7-(3-(isobutyryloxy)azetidin-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylate

442526-91-2